Recombinant CD40-ligand

CytokineRx: ResearchCompound: Investigational

Also known as: CD154, CD40 Ligand recombinant, CD40L, rCD154, rCD40L, TNFSF5, TRAP (TNF-Related Activation Protein)

Educational Only — Not medical advice. Consult a qualified clinician before using any peptide.

Source Recombinant CD40-ligand at Peptiology

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Summary

Recombinant soluble CD40‑ligand (CD154) is a biologic protein used experimentally to stimulate CD40‑mediated immune responses, investigated as a vaccine adjuvant and cancer immunotherapy.

Mechanism of Action

Soluble CD40 ligand binds CD40 on antigen‑presenting cells, triggering NF‑κB activation and enhancing immune cell activation

Routes of Administration

IntratumoralIntravenousSubcutaneous

Goals & Uses

  • Vaccine adjuvantVaccinologyModerate
  • Platelet activation researchHematology / ResearchModerate
  • Cancer immunotherapyOncologyModerate
  • B cell immunodeficiency (Hyper-IgM syndrome)Immunology / Rare DiseaseLow

Contraindications

  • History of thromboembolic eventsHematologicalHigh
  • Severe cardiovascular diseaseCardiovascularHigh
  • Active autoimmune diseaseAutoimmunityModerate

Adverse Effects

  • Cytokine release syndromeImmunologicUnknownSystemic inflammatory response from immune activation
  • Thromboembolic events (DVT, PE, arterial thrombosis)Hematological / VascularUncommon
  • Flu‑like symptomsSystemicUnknown
  • Injection site reactionsLocalCommon
  • Fever / flu-like symptomsSystemicCommon
  • Anti-drug antibody formationImmunologicalUncommon
  • Cytokine release / inflammatory responseImmunologicalUncommon

Drug Interactions

  • Antiplatelet agents (aspirin, clopidogrel)Low
  • Immunosuppressive agents (e.g., corticosteroids, cyclosporine)Moderate
  • Anticoagulants (warfarin, heparin, direct oral anticoagulants)Moderate

Population Constraints

  • Pediatric patientsAgeRelative
  • Patients with hypercoagulable statesHematologicalAbsolute
  • Pregnant or breastfeeding womenReproductiveAbsolute
  • Elderly patientsAgeRelative
  • Pregnant womenReproductiveRelative

Regulatory Status

  • European UnionInvestigationalUnder clinical investigation in Europe
  • United StatesInvestigationalInvestigational biologic; not FDA‑approved
  • United KingdomInvestigationalNo MHRA approval. Follows similar status to EU; no approved therapeutic use.

No approved indication in any major jurisdiction. Early-phase clinical trials were halted or suspended due to serious thromboembolic events. Remains primarily a research-stage molecule. Some investigational use continues in ex vivo settings and as a vaccine adjuvant component.

Evidence & Sources

No sources recorded yet.

Frequently Asked Questions

What is Recombinant CD40-ligand?

Recombinant soluble CD40‑ligand (CD154) is a biologic protein used experimentally to stimulate CD40‑mediated immune responses, investigated as a vaccine adjuvant and cancer immunotherapy.

What is Recombinant CD40-ligand used for?

Recombinant CD40-ligand is educationally associated with: Vaccine adjuvant, Platelet activation research, Cancer immunotherapy, B cell immunodeficiency (Hyper-IgM syndrome). Educational only — not medical advice.

How is Recombinant CD40-ligand administered?

Recorded routes of administration: Intratumoral, Intravenous, Subcutaneous.

What are the potential side effects of Recombinant CD40-ligand?

Reported adverse effects include: Cytokine release syndrome, Thromboembolic events (DVT, PE, arterial thrombosis), Flu‑like symptoms, Injection site reactions, Fever / flu-like symptoms, Anti-drug antibody formation, Cytokine release / inflammatory response. This list is not exhaustive — consult a qualified clinician.

Who should avoid Recombinant CD40-ligand?

Recorded contraindications: History of thromboembolic events, Severe cardiovascular disease, Active autoimmune disease. Consult a qualified clinician before use.

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